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Source comparison

What's the Half-Life of Tesamorelin: GHRH Analogue Comparison

Tesamorelin 26–43 minutes 2–3 hours Once daily GHRH receptor agonist with DPP-4 resistance Ideal for physiological pulsatile GH patterns without receptor desensitisation. Clinical data supports 52+ weeks continuous use Sermorelin 10–20 minutes 1.5–2 hours 1–2×

This comparison does not assign a generated winner or score.

  • Tesamorelin
  • 26–43 minutes
  • 2–3 hours
  • Once daily
  • GHRH receptor agonist with DPP-4 resistance
  • Ideal for physiological pulsatile GH patterns without receptor desensitisation. Clinical data supports 52+ weeks continuous use
  • Sermorelin
  • 10–20 minutes
  • 1.5–2 hours
  • 1–2× daily
  • GHRH receptor agonist, minimal DPP-4 resistance
  • Shorter action window requires more precise timing or split dosing; less forgiving than tesamorelin for meal proximity
  • CJC-1295 (no DAC)
  • 30 minutes
  • GHRH receptor agonist with extended stability
  • Functionally similar to tesamorelin; slightly longer half-life provides marginally wider injection window
  • CJC-1295 with DAC
  • 6–8 days
  • Sustained elevation
  • 1–2× weekly
  • GHRH receptor agonist with albumin binding
  • Convenient dosing but risks receptor downregulation and suppression of endogenous pulsatility with chronic use
  • GHRP-2
  • 20–30 minutes
  • 1–2 hours
  • 1–3× daily
  • Ghrelin receptor agonist
  • Often stacked with tesamorelin for synergistic GH release; acts on different pathway without extending half-life